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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T2120 | I-BET151 | GSK1210151A | Epigenetic Reader Domain |
I-BET151 (GSK1210151A) (GSK1210151A) is a specific BET inhibitor for BRD2/3/4 (IC50: 0.5/0.25/0.79 μM, in cell-free assays). | |||
T22845 | I-BET151 dihydrochloride | I-BET 151 hydrochloride | Others |
I-BET 151 dihydrochloride is a BET bromodomain inhibitor that prevents BET from recruiting to chromatin. |